Antagonist medications

Naltrexone vs Vivitrol.

Vivitrol is the monthly injection form of naltrexone — same medication, different formulation. How they compare, who fits which, and what to know about cost and induction.

Medically reviewed by N Elias, MD, board-certified in addiction medicine·Last reviewed May 2026
The short answer

Vivitrol is naltrexone. Specifically, Vivitrol is the brand name for the monthly intramuscular injection form of naltrexone. The daily pill form (sold as ReVia or generic naltrexone) and Vivitrol contain the same active medication — the difference is the formulation, the dosing interval, and how it’s given.

What is the difference between naltrexone and Vivitrol?

Both contain naltrexone, an opioid antagonist. Generic oral naltrexone is commonly used for alcohol use disorder and opioid blockade. Vivitrol is the extended-release injectable form FDA-approved for alcohol dependence and for prevention of return to use of opioid dependence after detoxification.

Vivitrol is naltrexone in a slow-release form — the same drug, packaged for monthly dosing instead of daily.

How do they compare?

FeatureOral naltrexoneVivitrol (injection)
Active medicationNaltrexoneNaltrexone
How it’s takenDaily pillMonthly intramuscular injection
Who administers itSelf at homeHealthcare provider in clinic
Adherence requirementDaily decisionOne decision per month
Typical cost without insuranceLower (generic available)Significantly higher
Telehealth-onlyPill can sometimes be prescribed by telehealth where legally permittedRequires in-person visit for the injection
Overdose risk after stoppingYes — opioid tolerance may be lower after stopping or missed dosesYes — especially near end of dosing interval, after a missed dose, or after stopping

Who fits each?

Oral naltrexone may be the better fit when:

Vivitrol may be the better fit when:

Both require an opioid-free period before starting

Whether daily or monthly, naltrexone requires a multi-day opioid-free interval before starting. Per Vivitrol labeling: at least 7–10 days off short-acting opioids; longer (often up to about 2 weeks) after methadone, buprenorphine, or other long-acting opioids. Starting too soon causes precipitated withdrawal — sudden, intense, and difficult to reverse.

There is no completely reliable way to know that every patient has had an adequate opioid-free interval; some clinicians use toxicology testing, clinical assessment, or a naloxone challenge when appropriate. Naltrexone labeling notes that no completely reliable method exists for determining whether a patient has had an adequate opioid-free period.

Once Vivitrol is given, the medication cannot simply be removed or stopped the way a pill can, and its antagonist effect persists across the monthly dosing interval — so precipitated withdrawal after a Vivitrol injection is harder to manage than after an oral dose.

Overdose risk if you stop and resume opioids. Naltrexone (in either form) reduces opioid tolerance. If treatment stops — whether intentionally or because a dose is missed — opioid use carries a higher overdose risk than before naltrexone. Vivitrol labeling specifically warns that the opioid blockade is surmountable, and that attempts to override the blockade with large amounts of opioids can lead to life-threatening intoxication or fatal overdose.

How much does Vivitrol cost?

Vivitrol is usually much more expensive than generic oral naltrexone. Actual cost depends on insurance, pharmacy or clinic billing, administration fees, manufacturer assistance, and site of care. Eligible patients may qualify for manufacturer (Alkermes) co-pay savings, subject to eligibility limits — ask the clinic that administers the injection about whether they participate.

Generic oral naltrexone is widely available and substantially less expensive than Vivitrol; check your local pharmacy or a discount program for a current cash price.

Medical sources
Medical note. This article is for education only and is not a substitute for medical advice. Medication choice, timing, dose changes, and stopping treatment should be handled with a licensed clinician. If you may be overdosing or having severe withdrawal, call 911 or seek emergency care.

See important safety information before use.

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